2010
Buděšínský M., Císařová I., Podlaha J., Borremans F. A. M., Martins J. C., Waroquier M., Pauwels E.:
Structures of cyclic dipeptides: an X-ray and computational study of cis- and trans-cyclo(Pip-Phe), cyclo(Pro-Phe) and their N-methyl derivatives.
Acta Crystallographica section B - Structural Science B66: 662-667, 2010.
Dračínský M., Pohl R., Slavětínská L., Buděšínský M.:
Observed and calculated 1H and 13C chemical shifts induced by the in situ oxidation of model sulfides to sulfoxides and sulfones.
Magnetic Resonance in Chemistry 48(9): 718-726, 2010.
Hlaváček J, Pícha J., Vaněk V., Jiráček J., Slaninová J., Fučík V., Buděšínský M., Gilner D., Holz R.C.:
Inhibitors of N (alpha)-acetyl-L-ornithine deacetylase: synthesis, characterization and analysis of their inhibitory potency.
Amino Acids 38(4): 1155-1164, 2010.
Karban J., Sýkora Jan., Kroutil J., Císařová I., Padělková Z., Buděšínský M.:
Synthesis of All Configurational Isomers of 1,6-Anhydro-2,3,4-trideoxy-2,3-epimino-4-fluoro-β-D-hexopyranoses.
Journal of Organic Chemistry 75(10): 3443-3446, 2010.
Kasal A, Buděšínský M., Griffiths W.J.:
Spectroscopic Methods of Steroid Analysis.
Steroid Analysis. Heidelberg : Springer, 2010 - (Malkin, H.; Gower, D.) 27-161. ISBN 978-1-4020-9774-4
Kočalka P., Rejman D., Vaněk V., Rinnová M., Tomečková I., Králíková Š., Petrová M., Páv O., Pohl R., Buděšínský M., Liboska R., Točík Z., Panova N., Votruba I., Rosenberg I.:
Structural diversity of nucleoside phosphonic acids as a key factor in the discovery of potent inhibitors of rat T-cell lymphoma thymidine phosphorylase.
Bioorganic and Medicinal Chemistry Letters 20(3): 862-865, 2010.
Kumprecht L., Buděšínský M., Bouř P., Kraus T.:
Alpha-cyclodextrins reversibly capped with disulfide bonds.
New Journal of Chemistry 34(10): 2254-2260, 2010.
Kvasnica M., Spáčilová P., Buděšínský M., Hajdúch M., Šarek, J.:
Oxidative cleavage of 3beta-acetoxy-21-oxolup-18-en-28-oic acid by ruthenium tetroxide.
Chemistry of Natural Compounds 46(4): 545-548, 2010.
Lepšík M., Srnec M., Plešek J., Buděšínský M., Klepetářová B., Hnyk D., Grüner B., Rulíšek L.:
Thiocyanation of closo-Dodecaborate B12H12 2-. A Novel Synthetic Route and Theoretical Elucidation of the Reaction Mechanism.
Inorganic Chemistry 49(11): 5040-5048, 2010.
Mojr V., Herzig V., Buděšínský M., Cibulka R., Kraus T.:
Flavin-cyclodextrin conjugates as catalysts of enantioselective sulfoxidations with hydrogen peroxide in aqueous media.
Chemical Communications 46(40): 7599-7601, 2010.
Monincová L., Buděšínský M., Slaninová J., Hovorka O., Cvačka J., Voburka Z., Fučík V., Borovičková L., Bednárová L., Straka M., Čeřovský V.:
Novel antimicrobial peptides from the venom of the eusocial bee Halictus sexcinctus (Hymenoptera: Halictidae) and their analogs.
Amino Acids 39(3): 763-775, 2010.
Niederhafner P., Bednárová L., Buděšínský M., Šafařík M., Ehala S., Ježek J., Borovičková L., Fučík V., Čeřovský V., Slaninová J.:
Melectin MAPs: the influence of dendrimerization on antimicrobial and hemolytic activity.
Amino Acids 39(5): 1553-1561, 2010.
Niederhafner P., Gut V., Ježek J., Buděšínský M., Kašička V., Wünsch E., Hlaváček J.:
Synthetic study on cystinyl peptides using solution and solid phase metodology: human IgG1 hinge region.
Amino Acids 39(3): 641-650, 2010.
Petrová M., Buděšínský M., Rosenberg I.:
Straightforward synthesis of 3´-deoxy-3´,4´-didehydronucleoside-5´-aldehydes via 2´,3´-O-orthoester group elimination: a simple route 3´,4´-didehydronucleosides.
Tetrahedron Letters 51(52): 6874-6876, 2010.
Pícha J., Buděšínský M., Fiedler P., Šanda M., Jiráček J.:
Synthesis of alpha-carboxyphosphinopeptides derived from norleucine.
Amino Acids 39(5): 1265-1280, 2010.
Pressová M., Buděšínský M., Kóšiová I., Kopecký V. Jr., Cvačka J., Kašička V., Šimák O., Točík Z., Rosenberg I.:
Oligomerization of adenosin-5´-O-ylmethylphosphonate, an isopolar AMP analogue: Evaluation of the route to short oligoadenylates.
Biopolymers 93(3): 277-289, 2010.
Šmidrkal J., Harmatha J., Buděšínský M., Vokáč K., Zídek Z., Kmoníčková E., Merkl R., Filip V.:
Modified approach for preparing (E)-stilbenes related to resveratrol, and evaluation of their potential immunobiological effects.
Collection of Czechoslovak Chemical Communications 75(2): 175-186, 2010.
Vaněk V., Pícha J., Buděšínský M., Šanda M., Jiráček J., Holz R. C., Hlaváček J.:
Synthesis of N-succinyl-L,L-diaminopimelic acid mimetics via selective protection.
Protein and Peptide Letters 17(3): 405-409, 2010.
Zelík P., Lukešová A., Čejka J., Buděšínský M., Havlíček V., Čegan A., Kopecký J.:
Nostotrebin 6, a bis(cyclopentenedione) with cholinesterase inhibitory activity isolated from Nostoc sp str. Lukesova 27/97.
Journal of Enzyme Inhibition and Medicinal Chemistry 25(3): 414-420, 2010.
Břehová P., Dračínský M., Holý A.:
Efficient Synthesis and Biological Properties of Base Substituted 2,4-Diamino-6-(R)-[3-hydroxy-2-(phosphonomethoxy)propoxy]pyrimidine (HPMPO-DAPy).
Antiviral Research 86(1): A52-A52, 2010.
Dračínský M., Bouř P.:
Computational analysis of solvent effects in NMR spectroscopy.
Journal of Chemical Theory and Computation 6(1): 288-299, 2010.
Dračínský M., Castaňo O., Kotora M., Bouř P.:
Rearrangement of Dewar Benzene Derivatives Studied by DFT.
Journal of Organic Chemistry 75(3): 576-581, 2010. .
Eignerová B., Janoušek Z., Dračínský M., Kotora J.:
Synthesis of Perfluoroalkylated Carboranes by Cross-Metathesis of Allylcarboranes and Perfluoroalkylpropenes.
Synlett 6(): 885-888, 2010.
Eignerová B., Sedlák D., Dračínský M., Bartůněk P., Kotora J.:
Synthesis and Biochemical Characterization of a Series of 17alpha-Perfluoroalkylated Estradiols as Selective Ligands for Estrogen Receptor alpha.
Journal of Medicinal Chemistry 53(19): 6947-6953, 2010.
Hocková D., Dračínský M., Holý A.:
Synthesis and Properties of a Novel Type of Acyclic Nucleoside Phosphonates: 2-(Purin-9-yl)ethoxyphenylphosphonic Acids.
European Journal of Organic Chemistry (15): 2885-2892, 2010.
Kapitán J., Dračínský M., Kaminský J., Benda L., Bouř P.:
Theoretical Modeling of Magnesium Ion Imprints in the Raman Scattering of Water.
Journal of Physical Chemistry B 114(10): 3574-3582, 2010.
Krečmerová M., Holý A., Andrei G., Pomeisl K., Tichý T., Břehová P., Masojídková M., Dračínský M., Pohl R., Laflamme G., Naesens L., Hui H., Cihlař T., Neyts J., De Clercq E., Balzarini J., Snoeck R.:
Synthesis of ester prodrugs of 9-(S)-[3-hydroxy-2-(phosphonomethoxy)propyl]-2,6-diaminopurine (HPMPDAP) as anti-poxvirus agents.
Journal of Medicinal Chemistry 53(19): 6825-6837, 2010.
Martínek V., Sklenář J., Dračínský M., Šulc M., Hofbauerová K., Bezouška K., Frei E., Stiborová M.:
Glycosylation protects proteins against free radicals generated from toxic xenobiotics.
Toxicological Sciences 117(2): 359-374, 2010.
Nencka R., Hřebabecký H., Dračínský M.:
Model synthesis of six-membered carbocyclic spironucleosides.
Collection of Czechoslovak Chemical Communications 75(12): 1259-1272, 2010.
Nencka R., Šála M., Dejmek M., Dračínský M., Holý A., Hřebabecký H.:
Two convergent approaches toward novel carbocyclic C-nucleosides.
Synthesis (23): 4119-4130, 2010.
Šála M., De Palma A. M., Hřebabecký H., Nencka R., Dračínský M., Leyssen P., Neyts J., Holý A.:
Design, synthesis, and biological evaluation of novel coxsackievirus B3 inhibitors.
Bioorganic & Medicinal Chemistry 18(12): 4374-4384, 2010.
Šála M., Hřebabecký H., Dračínský M., Masojídková M., De Palma A. M., Neyts J., Holý A.:
Synthesis of novel racemic carbocyclic nucleosides derived from 5,6-disubstituted norbornene.
Collection of Czechoslovak Chemical Communications 75(1): 1-20, 2010.
Čerňa I., Pohl R., Klepetářová B., Hocek M.:
Intramolecular Direct C-H Arylation Approach to Fused Purines. Synthesis of Purino[8,9-f]phenanthridines and 5,6-Dihydropurino[8,9-a]isoquinolines.
Journal of Organic Chemistry 75(7): 2302-2308, 2010.
Hasník Z., Pohl R., Hocek M.:
Synthesis of (Purin-6-yl)methylphosphonate Bases and Nucleosides.
Tetrahedron Letters 51(18): 2464-2466, 2010.
Ikonen S., Macíčková-Cahová H., Pohl R., Šanda M., Hocek M.:
Synthesis of nucleoside and nucleotide conjugates of bile acids, and polymerase construction of bile acid-functionalized DNA.
Organic & Biomolecular Chemistry 8(5): 1194-1201, 2010.
Janeba Z., Holý A., Pohl R., Snoeck R., Andrei G., De Clercq E., Balzarini J.:
Synthesis and biological evaluation of acyclic nucleotide analogues with a furo[2,3-d]pyrimidin-2(3H)-one base.
Canadian Journal of Chemistry 88(7): 628-638, 2010.
Khobragade D., Stensrud E. S., Mucha M., Smith J. R., Pohl R., Stibor I., Michl J.:
Preparation of Covalent Long-Chain Trialkylstannyl and Trialkylsilyl Salts and an Examination of their Adsorption on Gold.
Langmuir 26(11): 8483-8490, 2010.
Nauš P., Pohl R., Votruba I., Džubák P., Hajdúch M., Ameral R., Birkuš G., Wang T., Ray A. S., Mackman R., Cihlar T., Hocek M.:
6-(Het)aryl-7-Deazapurine Ribonucleosides as Novel Potent Cytostatic Agents.
Journal of Medicinal Chemistry 53(1): 460-470, 2010.
Raindlová V., Pohl R., Šanda M., Hocek M.:
Direct polymerase synthesis of reactive aldehyde-functionalized DNA and its conjugation and staining with hydrazines.
Angewandte Chemie. International Edition in English. 49(6): 1064-1066, 2010.
Spáčilová P., Nauš P., Pohl R., Votruba I., Snášel J., Zábranská H., Pichová I., Ameral R., Birkuš G., Cihlař T., Hocek M.:
CycloSal-Phosphate Pronucleotides of Cytostatic 6-(Het)aryl-7-Deazapurine Ribonucleosides: Synthesis, Cytostatic Activity, and Inhibition of Adenosine Kinases.
ChemMedChem 5(8): 1386-1396, 2010.
Synytsya A., Kim W. J., Kim S. M., Pohl R., Synytsya A., Kvasnička F., Čopíková J., Park Y. I.:
Structure and antitumour activity of fucoidan isolated from sporophyll of Korean brown seaweed Undaria pinnatifida.
Carbohydrate Polymers 81(1): 41-48, 2010.
Valášek M., Štursa J., Pohl R., Michl J.:
Lithium Salts of [1,12-Dialkyl-CB11Me10]- Anions.
Inorganic Chemistry 49(22): 10255-10263, 2010.
Valášek M., Štursa J., Pohl R., Michl J.:
Microwave-Assisted Alkylation of [CB11H12]- and Related Anions.
Inorganic Chemistry 49(22): 10247-10254, 2010.
Bárta J., Slavětínská L., Klepetářová B., Hocek M.:
Modular Synthesis of 5-Substituted Furan-2-yl C-2'-Deoxyribonucleosides and Biaryl Covalent Base-pair Analogues.
European Journal of Organic Chemistry (28): 5432-5443, 2010.
Kubelka T., Slavětínská L., Klepetářová B., Hocek M.:
Synthesis of 2,4-Disubstituted Pyrimidin-5-yl C-2'-Deoxyribonucleosides by Sequential Regioselective Reactions of 2,4-Dichloropyrimidine Nucleosides.
European Journal of Organic Chemistry (14): 2666-2669, 2010.
Štefko M., Slavětínská L., Klepetářová B., Hocek M.:
A General and Efficient Synthesis of Pyridin-2-yl C-Ribonucleosides Bearing Diverse Alkyl, Aryl, Amino and Carbamoyl Groups in Position 6.
Journal of Organic Chemistry 75(2): 442-449, 2010.
Kovalová A., Ledvina M., Šaman D., Zyka D., Kubíčková M., Žídek L., Sklenář V., Pompach P., Kavan D., Bílý J., Vaněk O., Kubínková Z., Libigerová M., Ivanová L., Antolíková M., Mrázek H., Rozbeský D., Hofbauerová K., Křen V., Bezouška K.:
Synthetic N-Acetyl-D-glucosamine Based Fully Branched Tetrasaccharide, a Mimetic of the Endogenous Ligand for CD69, Activates CD69+ Killer Lymphocytes upon Dimerization via a Hydrophilic Flexible Linker.
Journal of Medicinal Chemistry 53(10): 4050-4065, 2010.
Severa L., Adriaenssens L., Vávra J., Šaman D., Císařová I., Fiedler P., Teplý F.:
Highly modular assembly of cationic helical scaffolds: rapid synthesis of diverse helquats via differential quaternization.
Tetrahedron 66(19): 3537-3552, 2010.
Severa L., Koval D., Novotná P., Ončák M., Sázelová P., Šaman D., Slavíček P., Urbanová M., Kašička V., Teplý F.:
Resolution of a configurationally stable [5]helquat. enantiocomposition analysis of a helicene congener by capillary electrophoresis.
New Journal of Chemistry 34(6): 1063-1067, 2010.
Songis O., Míšek J., Schmid M. B., Kollárovič A., Stará I., Šaman D., Císařová I., Starý I.:
A Versatile Synthesis of Functionalized Pentahelicenes.
Journal of Organic Chemistry 75(20): 6889-6899, 2010.
Svobodová H., Ryšavá H., Pavlík M., Šaman D., Drašar P., Wimmer Z.:
Steroid conjugates: Synthesis and preliminary biological testing of pro-juvenoids.
Bioorganic & Medicinal Chemistry 18(23): 8194-8203, 2010.