2011
Čechová, L., Jansa, P., Šála, M., Dračínský, M., Holý, A., Janeba, Z.:
The optimized microwave-assisted decomposition of formamides
and its synthetic utility in the amination reactions of purines.
Tetrahedron 67: 866-871, 2011.
Dračínský, M., Jansa, P., Chocholoušová, J., Vacek, J., Kovačková, S., Holý, A.:
Mechanism of the isotopic exchange reaction of the 5-H hydrogen of uracil derivatives in water and
nonprotic solvents.
European Journal of Organic Chemistry 4: 777–785, 2011.
Dračínský, M., Jansa, P., Buděšínský, M.:
Tautomerism and the Protonation/Deprotonation of Isocytosine in Liquid- and Solid-States Studied
by NMR Spectroscopy and Theoretical Calculations.
European Journal of Organic Chemistry 8: 1544-1551, 2011.
Baszczyňski, O., Jansa, P., Dračínský, M., Klepetářová, B., Holý, A., Votruba, I.,
De Clercq, E., Balzarini, J., Janeba, Z.:
Synthesis and antiviral activity of N9-[3-fluoro-2-(phosphonomethoxy)propyl] analogues derived
from N6-substituted adenines and 2,6-diaminopurines.
Bioorg. Med. Chem. 19: 2114-2124, 2011.
Sedláček, O., Břehová, P., Pohl, R., Holý, A., Janeba, Z.:
The synthesis of the 8-C-substituted 2,6-diamino-9-[2-(phosphonomethoxy)ethyl]purine (PMEDAP) derivatives by
diverse cross-coupling reactions.
Can. J. Chem. 89: 488-498, 2011.
Jansa, P., Holý, A., Dračínský, M., Baszczyňski, O., Česnek, M., Janeba, Z.:
Efficient and 'green' microwave-assisted synthesis of haloalkylphosphonates via the Michaelis-Arbuzov reaction.
Green Chem. 13: 882-888, 2011.
Jirásková-Vanícková, J., Ettrich, R., Vorlová, B., Hoffman, H. E., Lepšík, M., Jansa, P., Konvalinka, J.:
Inhibition of Human Serine Racemase, an Emerging Target for Medicinal Chemistry.
Curr. Drug Targets 12: 1037-1055, 2011.
Hocková, D., Holý, A., Andrei, G., Snoeck, R., Balzarini, J.:
Acyclic nucleoside phosphonates with a branched 2-(2-phosphonoethoxy)ethyl
chain: Efficient synthesis and antiviral activity.
Bioorg. Med. Chem. 19: 4445-4453, 2011.
Jersey, J., Holy, A., Hockova, D., Naesens, L., Keough, D. T., Guddat, L. W.:
6-Oxopurine Phosphoribosyltransferase: A Target for the Development of Antimalarial Drugs.
Current Topics in Medicinal Chemistry 11: 2085-2102, 2011.
Jansa, P., Votruba, I., Břehová, P., Dračínský, M., Klepetářová, B., Janeba, Z.:
Efficient one-pot synthesis of polysubstituted 6-[(1H-1,2,3-triazol-1-yl)methyl]uracils through the "click" protocol.
Collect. Czech. Chem. Commun. 76: 1121-1131, 2011.
Břehová, P., Česnek, M., Dračínský, M., Holý, A., Janeba, Z.:
The efficient synthesis of 2-arylpyrimidine acyclic nucleoside phosphonates using Liebeskind-Srogl cross-coupling reaction.
Tetrahedron 67: 7379-7385, 2011.
Jansa, P., Baszczyňski, O., Dračínský, M., Votruba, I., Zídek, Z., Bahador, G., Stepan, G., Cihlar, T., Mackman, R.,
Holý, A., Janeba, Z.:
A novel and efficient one-pot synthesis of symmetrical diamide (bis-amidate) prodrugs of acyclic nucleoside phosphonates and evaluation of
their biological activities.
Eur. J. Med. Chem. 46: 3748-3754, 2011.