2013

Jansa, P., Čechová, L.; Dračínský, M., Janeba, Z.:
A conversion of aromatic thiocyanates into sulfothioates: new synthetic route to aromatic Bunte salts.
RSC Advances 3: 1282-1284, 2013.
 
Keough, D. T., Špaček, P., Hocková, D., Tichý, T., Vrbková, S., Slavětínská, L., Janeba, Z., Naesens, L., Edstein, M. D., Chavchich, M., Wang, T.-H., de Jersey, J., Guddat, L. W.:
Acyclic nucleoside phosphonates containing a second phosphonate group are potent inhibitors of 6-oxopurine phosphoribosyltransferases and have antimalarial activity.
Journal of Medicinal Chemistry 56: 2513-2526, 2013.
 
Dolečková, I., Česnek, M., Dračínský, M., Brynda, J., Voller, J., Janeba, Z., Kryštof, V.:
Synthesis and biological evaluation of guanidino analogues of roscovitine.
European Journal of Medicinal Chemistry 62: 443-452, 2013.
 
Krečmerová, M., Jansa, P., Dračínský, M., Sázelová, P., Kašička, V., Neyts, J., Auwerx, J., Kiss, E., Goris, N., Stepan, G., Janeba, Z.:
9-[2-(R)-(Phosphonomethoxy)propyl]-2,6-diaminopurine (R)-PMPDAP and its prodrugs: Optimized preparation, including identification of by-products formed, and antiviral evalution in vitro.
Bioorganic & Medicinal Chemistry 2013, 21, 1199-1208.
 
Baszczyňski, O., Hocková, D., Janeba, Z., Holý, A.; Jansa, P.; Dračínský, M., Keough, D. T., J., Guddat, L. W.:
The effect of novel [3-fluoro-(2-phosphonoethoxy)propyl]purines on the inhibition of Plasmodium falciparum, Plasmodium vivax and human hypoxanthine-guanine-(xanthine) phosphoribosyltransferases.
European Journal of Medicinal Chemistry 67: 81-89, 2013.

Mandíková, J., Volková, M., Pávek, P., Česnek, M., Janeba, Z., Kubíček, V., Trejtnar, F.: Interactions with selected drug renal transporters and transporter-mediated cytotoxicity in antiviral agents from the group of acyclic nucleoside phosphonates.
Toxicology 311: 135-146, 2013.
 

Keough, D. T., Hocková, D., Rejman, D., Špaček, P., Vrbková, S., Krečmerová, M., Soon Eng, W., Jans, H., West, N. P., Naesens, L. M. J., de Jersey, J., Guddat, L. W.: Inhibition of the Escherichia coli 6-oxopurine phosphoribosyltransferases by nucleoside phosphonates: Potential for new antibacterial agents.
Journal of Medicinal Chemistry 56: 6967-6984, 2013.