2014

Milan Dejmek, Michal Šála, Pavla Plačková, Hubert Hřebabecký, Laura Mascarell, Johan Neyts, Martin Dračínský, Eliška Procházková, Petr Jansa, Pieter Leyssen, Helena Mertlíková-Kaiserová and Radim Nencka:
Synthesis of Novel Purine-Based Coxsackievirus Inhibitors Bearing Polycylic Substituents at the N-9 Position
Archiv der Pharmazie 347: 478-485, 2014.

Radim Nencka, Hubert Hřebabecký, Michal Šála and Milan Dejmek:
Nízkomolekulární inhibitoty replikace enterovirů
Chemické Listy 108: 326-334, 2014.

Milan Dejmek, Hubert Hřebabecký, Michal Šála, Martin Dračínský, Eliška Procházková, Pieter Leyssen, Johan Neyts, Jan Balzarini and Radim Nencka:
From norbornane-based nucleotide analogs locked in South conformation to novel inhibitors of feline herpes virus
Bioorganic & Medicinal Chemistry 22: 2974-2983, 2014.

Pavla Plačková, Hubert Hřebabecký, Michal Šála, Radim Nencka, Tomáš Elbert, and Helena Mertlíková-Kaiserová:
Transport mechanisms of a novel antileukemic and antiviral compound 9-norbornyl-6-chloropurine
Journal of Enzyme Inhibition and Medicinal Chemistry in press.

Martin Dračínský, Michal Šála and Paul Hodgkinson:
Dynamics of water molecules and sodium ions in solid hydrates of nucleotides
CrystEngComm 16: 6756-6764, 2014.

Lucia Kučerová, Lucia Feketeová, Zuzana Kozovská, Martina Poturnajová, Miroslava Matušková, Radim Nencka and Pavel Babal:
In Vivo 5FU-Exposed Human Medullary Thyroid Carcinoma Cells Contain a Chemoresistant CD133+ Tumor–Initiating Cell Subset
Thyroid 24(3): 520-532, 2014.

Adriana Baumlová, Dominika Chalupská, Bartosz Róźycki, Marko Jovic, Eva Wisniewski, Martin Klíma, Anna Dubánková, Daniel P. Kloer, Radim Nencka, Tamas Balla and Evžen Bouřa:
The crystal structure of the phosphatidylinositol 4-kinase IIα
EMBO reports 15: 1085-1092, 2014.

Jakub Šebera, Lukáš Trantírek, Yoshiuki Tanaka, Radim Nencka, Jiří Fukal and Vladimír Sychrovský:
The activation of N-glycosidic bond cleavage operated by base-excision repair enzyme hOGG1; theoretical study of the role of Lys 249 residue in activation of G, OxoG and FapyG
RSC Advances 4: 44043-44051, 2014.

Milan Dejmek, Michal Šála, Hubert Hřebabecký, Martin Dračínský, Eliška Procházková, Dominika Chalupská, Martin Klíma, Pavla Plačková, Miroslav Hájek, Graciela Andrei, Lieve Naesens, Pieter Leyssen, Johan Neyts, Jan Balzarini, Evžen Bouřa, and Radim Nencka:
Norbornane-based nucleoside and nucleotide analogues locked in North conformation
Bioorganic & Medicinal Chemistry 2014 in press.