2012

Česnek M., Hocková D., Holý A., Dračínský M., Baszczyňski O., de Jersey J., Keough D.T., Guddat L.W.:
Synthesis of 9-phosphonoalkyl and 9-phosphonoalkoxyalkyl purines: Evaluation of their ability to act as inhibitors of Plasmodium falciparum, Plasmodium vivax and human hypoxanthine-guanine-(xanthine) phosphoribosyltransferases.
Bioorganic and Medicinal Chemistry 20: 1076-1089, 2012.

Krečmerová M., Dračínský M., Hocková D., Holý A., Keough D.T., Guddat L.W.:
Synthesis of purine N9-[2-hydroxy-3-O-(phosphonomethoxy)propyl] derivatives and their side-chain modified analogues as potential antimalarial agents.
Bioorganic and Medicinal Chemistry 20: 1222-1230, 2012.

Jansa P., Hradil O., Baszczyňski O., Dračínský M., Klepetářová B., Holý A., Balzarini J., Janeba Z.:
An efficient microwave-assisted synthesis and biological properties of polysubstituted pyrimidinyl- and 1,3,5-triazinylphosphonic acids.
Tetrahedron 68: 865-871, 2012.

Baszczyňski O., Jansa P., Dračínský M., Kaiser M.M., Špaček P., Janeba Z.:
An efficient oxa-Michael addition to diethyl vinylphosphonate under mild reaction conditions.
RSC Advances 2: 1282-1284, 2012.

Procházková E., Jansa P., Dračínský M., Holý A., Mertlíková-Kaiserová H.:
Determination of the antioxidative activity of substituted 5-aminopyrimidines.
Free Radical Research 46: 61-67, 2012.

Kaiser M.M., Jansa P., Dračínský M., Janeba Z.:
A novel type of acyclic nucleoside phosphonates derived from 2-(phosphonomethoxy)propanoic acid.
Tetrahedron 68: 4003-4012, 2012.

Jansa P., Baszczyňski O., Procházková E., Dračínský M., Janeba Z.:
Microwave-assisted hydrolysis of phosphonate diesters: An efficient protocol for the preparation of phosphonic acids.
Green Chemistry 14: 2282-2288, 2012.

Hocková D., Keough D.T., Janeba Z., Wang T.-H., de Jersey J., Guddat L.W.:
Synthesis of novel N-branched acyclic nucleoside phosphonates as potent and selective inhibitors of human, Plasmodium falciparum and Plasmodium vivax 6-oxopurine phosphoribosyltransferases.
Journal of Medicinal Chemistry 55: 6209-6223, 2012.