2017

Kolman V., Jansa P., Kalčic F., Janeba Z.*, Zídek Z.*:
Polysubstituted 4,6-bis(hetero)arylpyrimidines as dual inhibitors of nitric oxide and prostaglandin E2 production.
Nitric Oxide 67: 53–57, 2017.

Kaiser M.M., Baszczyňski O., Hocková D., Poštová-Slavětínská L., Dračínský M., Keough D.T., Guddat L.W., Janeba Z.*:
Acyclic nucleoside phosphonates containing 9-deazahypoxanthine and a five-membered heterocycle as selective inhibitors of plasmodial 6-oxopurine phosphoribosyltransferases.
ChemMedChem 12: 1133–1141, 2017.

Lukáč M., Hocková D., Keough D.T., Guddat L.W., Janeba Z.:
Novel nucleotide analogues bearing (1H-1,2,3-triazol-4-yl)phosphonic acid moiety as inhibitors of Plasmodium and human 6-oxopurine phosphoribosyltransferases.
Tetrahedron 73: 692-702, 2017.

Eng W.S., Keough D.T., Hocková D., Winzor D.J., Guddat L.W.:
Oligomeric state of hypoxanthine-guanine phosphoribosyltransferase from Mycobacterium tuberculosis.
Biochimie 135: 6-14, 2017.

Špaček P., Keough D.T., Chavchichc M., Dračínský M., Janeba Z., Naesens L., Edstein M.D., Guddat L.W., Hocková D.*:
Synthesis and evaluation of symmetric acyclic nucleoside bisphosphonates as inhibitors of the Plasmodium falciparum, Plasmodium vivax and human 6-oxopurine phosphoribosyltransferases and the antimalarial activity of their prodrugs.
Bioorganic & Medicinal Chemistry 25: 4008–4030, 2017.