2016

Eng W.S., Hocková D.*, Špaček P., Baszczyňski O., Janeba Z., Naesens L., Keough D.T., Guddat L.W.*:
Crystal Structures of Acyclic Nucleoside Phosphonates in Complex with Escherichia coli Hypoxanthine Phosphoribosyltransferase.
ChemistrySelect 1: 6267-6276, 2016.

Břehová P., Šmídková M., Skácel J., Dračínský M., Mertlíková-Kaiserová H., Soto Velasquez M.P., Watts V.J., Janeba Z.:
Design and synthesis of fluorescent acyclic nucleoside phosphonates as potent inhibitors of bacterial adenylate cyclases.
ChemMedChem 11: 2534–2546, 2016.

Terán D., Hocková D., Česnek M., Zíková A., Naesens L., Keough D.T., Guddat L.W.:
Crystal structures and inhibition of Trypanosoma brucei hypoxanthine–guanine phosphoribosyltransferase.
Scientific Reports 6: 35894, 2016.

Procházková E., Čechová L., Tarábek J., Janeba Z.*, Dračínský M.*:
Tunable Push–Pull Interactions in 5-Nitrosopyrimidines.
Journal of Organic Chemistry 81: 3780-3789, 2016.

Kaiser M.M., Poštová-Slavětínská L., Dračínský M., Lee Y.J., Tian Y., Janeba Z.:
Synthesis and biological properties of prodrugs of (S)-3-(adenin-9-yl)-2-(phosphonomethoxy)propanoic acid.
European Journal of Medicinal Chemistry 108: 374-380, 2016.

Mandíková J., Volková M., Pávek P., Navrátilová L., Hyršová L., Janeba Z., Pavlík J., Bárta P., Trejtnar F.:
Entecavir interacts with influx transporters hOAT1, hCNT2, hCNT3, but not with hOCT2: The potential for renal transporter-mediated cytotoxicity and drug-drug interactions.
Frontiers in Pharmacology 6: 1-11, 2016.

Šolínová V., Mikysková H., Kaiser M.M., Janeba Z., Holý A., Kašička V.:
Estimation of apparent binding constant of complexes of selected acyclic nucleoside phosphonates with ß-cyclodextrin by affinity capillary electrophoresis.
Electrophoresis 37: 239-247, 2016.

Zouharová D., Lipenská I., Fojtíková M., Kulich P., Neca J., Slaný M., Kovarčík K., Turánek-Knotigová P., Hubatka F., Čelechovská H., Mašek J., Koudelka S., Procházka L., Eyer L., Plocková J., Bartheldyová E., Miller A.D., Růžek D., Raška M., Janeba Z., Turánek J.:
Antiviral activities of 2,6-diaminopurine-based acyclic nucleoside phosphonates against herpesviruses: In vitro study results with pseudorabies virus (PrV, SuHV-1).
Veterinary Microbiology 184: 84-93, 2016.

Špak J., Janeba Z., Jansa P., Baszczyňski O., Pavingerová D., Špaková V.:
Phytotoxicity of acyclic nucleoside phosphonates in Brassica pekinensis and Solanum lycopersicum.
Plant Cell, Tissue and Organ Culture 125: 375-379, 2016.

Zídek Z., Kverka M., Dusilová A., Kmoníčková E., Jansa P.:
Dual inhibition of nitric oxide and prostaglandin E2 production by polysubstituted 2-aminopyrimidines.
Nitric oxide 57: 48-56, 2016.

Šimon P., Baszczyňski O., Šaman D., Stepan G., Hu E., Lansdon E.B., Jansa P., Janeba, Z.:
Novel (2,6-difluorophenyl)(2-(phenylamino)pyrimidin-4-yl) methanones with restricted conformation as potent non-nucleoside reverse transcriptase inhibitors against HIV-1.
European Journal of Medicinal Chemistry 122: 185-195, 2016.