2010

Janeba, Z., Masojídková, M., Holý, A.:
Alternative synthesis of 9-{3-[(diisopropoxyphosphoryl)methoxy]-2-hydroxypropyl}adenine and its free phosphonates substituted at the C-8 position of purine base.
Collection of Czechoslovak Chemical Communications 75: 371-381, 2010.

Hocková, D., Dračínský, M., Holý, A.:
Synthesis and properties of a novel type of acyclic nucleoside phosphonates: 2-(Purin-9-yl)ethoxyphenylphosphonic acids.
European Journal of Organic Chemistry 15: 2885-2892, 2010.

Janeba, Z., Holý, A., Pohl, R., Snoeck, R., Andrei, G., De Clercq, E., Balzarini, J.:
Synthesis and biological evaluation of acyclic nucleotide analogues with a furo[2,3-d]pyrimidin-2(3H)-one base.
Can. J. Chem. 88: 628-638, 2010.

Keough, D. T., Hocková, D., Krečmerová, M., Česnek, M., Holý, A., Naesens, L., Brereton, I. M., Winzor, D. J., de Jersey, J., Guddat, L. W.:
Plasmodium vivax hypoxanthine-guanine phosphoribosyltransferase: A target for anti-malarial chemotherapy.
Mol. Biochem. Parasitol. 173: 165-169, 2010.

Elbert, T., Břehová, P., Holý, A.:
The preparation of 3H-labeled acyclic nucleoside phosphonates and study of their stability.
Collection of Czechoslovak Chemical Communications 75: 757-766, 2010.

Krečmerová, M., Holý, A., Andrei, G., Pomeisl, K., Tichý, T., Břehová, P., Masojídková, M., Dračínský, M., Pohl, R., Laflamme, G., Naesens, L., Hui, H., Cihlar, T., Neyts, J., De Clercq, E., Balzarini, J., Snoeck, R.:
Synthesis of ester prodrugs of 9-(S)-[3-hydroxy-2-(phosphonomethoxy)propyl]-2,6-diaminopurine (HPMPDAP) as anti-poxvirus agents.
J. Med. Chem. 53: 6825-6837, 2010.

Votruba, I., Trýznová, J., Břehová, P., Tloušťová, E., Horská, K.,Fanfrlík, J., Přenosil, O., Holý, A.:
Inhibition of human purine nucleoside phosphorylase by tenofovir phosphate congeners.
Collection of Czechoslovak Chemical Communications 75: 1249-1257, 2010.

Česnek, M., Herdewijn, P.:
Synthesis and anti-HIV activity of new 3'-O-phosphonomethyl nucleosides.
Heterocycles 82: 663-687, 2010.