2018
Čechová L., Kind J., Dračínský M., Filo J., Janeba Z., Thiele C. M., Cigáň M., Procházková E.:
Photoswitching behaviour of 5-phenylazopyrimidines: in situ irradiation NMR and optical spectroscopy combined with theoretical methods.
Journal of Organic Chemistry 83: 5986–5998, 2018.
Kolman V., Kalčic F., Jansa P., Zídek Z.,* Janeba Z.:*
Influence of the C-5 substitution in polysubstituted pyrimidines on inhibition of prostaglandin E2 production.
European Journal of Medicinal Chemistry 156: 295–301, 2018.
Kaiser M.M., Novák P., Rosenbergová Š., Poštová-Slavětínská L., Rosenberg I.,* Janeba Z.:*
Acyclic nucleoside phosphonates bearing (R)- or (S)-9-[3-hydroxy-2-(phosphonoethoxy)propyl] (HPEP) moiety as monomers for the synthesis of modified oligonucleotides.
European Journal of Organic Chemistry 5119–5126, 2018.
Česnek M., Skácel J., Jansa P., Dračínský M., Šmídková M., Mertlíková-Kaiserová H., Soto-Velasquez M. P., Watts V. J.,* Janeba Z.:*
Nucleobase modified adefovir (PMEA) analogues as potent and selective inhibitors of adenylate cyclases from Bordetella pertussis and Bacillus anthracis.
ChemMedChem 13: 1779–1796, 2018.
Bray M., Andrei G., Ballana E., Carter K., Durantel D., Gentry B., Janeba Z., Moffat J., Oomen C.J., Tarbet B., Riveira-Muñoz E., Esté J.A.:
Meeting report: 31st International Conference on Antiviral Research.
Antiviral Research 158: 88–102, 2018.
Štěpánová S., Procházková E., Čechová L., Žurek J., Janeba Z., Dračínský M., Kašička V.:
Separation of rotamers of 5-nitrosopyrimidines and estimation of binding constants of their complexes with β-cyclodextrin by capillary electrophoresis.
Journal of Chromatography A 1570: 164–171, 2018.
Klejch T., Pohl R., Janeba Z., Sun M., Keough D.T., Guddat L.W.*, Hocková D.*:
Acyclic nucleoside phosphonates with unnatural nucleobases, favipiravir and allopurinol, designed as potential inhibitors
of the human and Plasmodium falciparum 6-oxopurine phosphoribosyltransferases.
Tetrahedron 74: 5886-5897, 2018.
Procházková E., Čechová L., Kind J., Janeba Z., Thiele C.M., Dračínský M.:
Photoswitchable intramolecular hydrogen bonds in 5-phenylazopyrimidines revealed by in situ irradiation NMR spectroscopy.
Chemistry - A European Journal 24: 492–498, 2018.
Frydrych J., Skácel J., Šmídková M., Mertlíková-Kaiserová H., Dračínský M., Gnanasekaran R., Lepšík M., Soto-Velasquez M., Watts V.J., Janeba Z.:
Synthesis of α-branched acyclic nucleoside phosphonates as potential inhibitors of bacterial adenylate cyclases.
ChemMedChem 13: 199–206, 2018.
Keough D.T., Rejman D.,* Pohl R., Zborníková E., Hocková D., Croll T., Edstein M.D., Birrell G.W., Chavchich M., Naesens L.M.J., Pierens G.K.,
Brereton I.M., Guddat L.W.:
The Design of Plasmodium vivax Hypoxanthine-Guanine Phosphoribosyltransferase Inhibitors as Potential Antimalarial Therapeutics.
ACS Chemical Biology 13: 82-90, 2018.
Doleželová E., Teran D., Gahura O., Kotrbová Z., Procházková M., Keough D., Špaček P., Hocková D., Guddat L., Zíková A.:
Evaluation of the Trypanosoma brucei 6-oxopurine salvage pathway as a potential target for drug discovery.
PLOS Neglected Tropical Diseases 12 (2): e0006301, 2018.